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Neddylation inhibitor MLN4924 suppresses growth and migration of human gastric cancer cells

MLN4924 is a recently discovered small molecule inhibitor of NEDD8-Activating Enzyme (NAE). Because cullin RING ligase (CRL), the largest family of E3 ubiquitin ligase, requires cullin neddylation for its activity, MLN4924, therefore, acts as an indirect inhibitor of CRL by blocking cullin neddylati...

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Pubblicato in:Sci Rep
Autori principali: Lan, Huiyin, Tang, Zaiming, Jin, Hongchuan, Sun, Yi
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4827092/
https://ncbi.nlm.nih.gov/pubmed/27063292
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep24218
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