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Covalent Bonding of Pyrrolobenzodiazepines (PBDs) to Terminal Guanine Residues within Duplex and Hairpin DNA Fragments

Pyrrolobenzodiazepines (PBDs) are covalent-binding DNA-interactive agents with growing importance as payloads in Antibody Drug Conjugates (ADCs). Until now, PBDs were thought to covalently bond to C2-NH(2) groups of guanines in the DNA-minor groove across a three-base-pair recognition sequence. Usin...

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Bibliografiska uppgifter
I publikationen:PLoS One
Huvudupphovsmän: Mantaj, Julia, Jackson, Paul J. M., Karu, Kersti, Rahman, Khondaker M., Thurston, David E.
Materialtyp: Artigo
Språk:Inglês
Publicerad: Public Library of Science 2016
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC4824457/
https://ncbi.nlm.nih.gov/pubmed/27055050
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0152303
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