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Engineered kinesin motor proteins amenable to small-molecule inhibition

The human genome encodes 45 kinesin motor proteins that drive cell division, cell motility, intracellular trafficking and ciliary function. Determining the cellular function of each kinesin would benefit from specific small-molecule inhibitors. However, screens have yielded only a few specific inhib...

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Pubblicato in:Nat Commun
Autori principali: Engelke, Martin F., Winding, Michael, Yue, Yang, Shastry, Shankar, Teloni, Federico, Reddy, Sanjay, Blasius, T. Lynne, Soppina, Pushpanjali, Hancock, William O., Gelfand, Vladimir I., Verhey, Kristen J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4822052/
https://ncbi.nlm.nih.gov/pubmed/27045608
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/ncomms11159
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