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Molecular imaging of EGFR and CD44v6 for prediction and response monitoring of HSP90 inhibition in an in vivo squamous cell carcinoma model

PURPOSE: Heat shock protein 90 (HSP90) is essential for the activation and stabilization of numerous oncogenic client proteins. AT13387 is a novel HSP90 inhibitor promoting degradation of oncogenic proteins upon binding, and may also act as a radiosensitizer. For optimal treatment there is, however,...

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Detalhes bibliográficos
Publicado no:Eur J Nucl Med Mol Imaging
Main Authors: Spiegelberg, Diana, Mortensen, Anja C., Selvaraju, Ram K., Eriksson, Olof, Stenerlöw, Bo, Nestor, Marika
Formato: Artigo
Idioma:Inglês
Publicado em: Springer Berlin Heidelberg 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4819754/
https://ncbi.nlm.nih.gov/pubmed/26627081
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00259-015-3260-x
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