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An Asymmetric Vinylogous Michael Cascade of Silyl Glyoximide, Vinyl Grignard, and Nitroalkenes via Long Range Stereoinduction

A diastereoselective auxiliary-mediated vinylation/[1,2]-Brook rearrangement/vinylogous Michael cascade of silyl glyoximide, vinylmagnesium bromide, and nitroalkenes is described. The reaction occurs with complete regio- and diastereocontrol in good yield. The diastereoselectivity is induced by a ra...

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Detalhes bibliográficos
Publicado no:J Org Chem
Main Authors: Boyce, Gregory R., Johnson, Jeffrey S.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4761320/
https://ncbi.nlm.nih.gov/pubmed/26833255
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.joc.5b02693
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