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A bead-based proximity assay for BRD4 ligand discovery

Bromodomain-containing proteins have emerged as desirable targets for anti-neoplastic and anti-inflammatory drug discovery. Toward the development of selective inhibitors of the BET family of bromodomains, we optimized bead-based assays to detect interactions between bromodomains and poly-acetylated...

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Detalhes bibliográficos
Publicado no:Curr Protoc Chem Biol
Main Authors: Roberts, Justin M., Bradner, James E.
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4725578/
https://ncbi.nlm.nih.gov/pubmed/26629616
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/9780470559277.ch150024
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