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Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation

Signal Transducer and Activator of Transcription 5 (STAT5) protein, a component of the STAT family of signaling proteins, is considered to be an attractive therapeutic target because of its involvement in the progression of acute myeloid leukemia. In an effort to discover potent molecules able to in...

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Vydáno v:Eur J Med Chem
Hlavní autoři: Romagnoli, Romeo, Baraldi, Pier Giovanni, Prencipe, Filippo, Lopez-Cara, Carlota, Rondanin, Riccardo, Simoni, Daniele, Hamel, Ernest, Grimaudo, Stefania, Pipitone, Rosaria Maria, Meli, Maria, Tolomeo, Manlio
Médium: Artigo
Jazyk:Inglês
Vydáno: 2015
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4724257/
https://ncbi.nlm.nih.gov/pubmed/26629859
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2015.11.022
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