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Novel (64)Cu-Radiolabeled Bile Acid Conjugates for Targeted PET Imaging

A promising bifunctional chelate (N-NE3TA) was conjugated to bile acids, cholic acid (CA), deoxycholic acid (DCA), and chenodeoxycholic acid (CDCA) as tumor targeting vectors. Bile acid conjugates of N-NE3TA (CA-N-NE3TA, DCA-N-NE3TA, and CDCA-N-NE3TA) were comparatively evaluated for complexation wi...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Main Authors: Chong, Hyun-Soon, Chen, Yunwei, Kang, Chi Soo, Sun, Xiang, Wu, Ningjie
Formato: Artigo
Idioma:Inglês
Publicado: 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4706377/
https://ncbi.nlm.nih.gov/pubmed/25661712
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.01.008
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