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Whacking a mole-cule: clinical activity and mechanisms of resistance to third generation EGFR inhibitors in EGFR mutated lung cancers with EGFR-T790M

Epidermal growth factor receptor (EGFR) mutations, especially EGFR-exon 19 deletions and EGFR-L858R, are the most frequent actionable genomic events in lung adenocarcinomas. Tumors arise due to constitutively activated EGFR signaling and are susceptible to EGFR tyrosine kinase inhibitors (TKIs). Fir...

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Dettagli Bibliografici
Pubblicato in:Transl Lung Cancer Res
Autori principali: Costa, Daniel B., Kobayashi, Susumu S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: AME Publishing Company 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4700227/
https://ncbi.nlm.nih.gov/pubmed/26798593
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3978/j.issn.2218-6751.2015.05.05
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