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Iminoboronate Formation Leads to Fast and Reversible Conjugation Chemistry of α-Nucleophiles at Neutral pH

Bioorthogonal reactions that are fast and reversible under physiologic conditions are in high demand for biological applications. Herein, we show that an ortho boronic acid substituent makes aryl ketones to rapidly conjugate with α-nucleophiles at neutral pH. Specifically, 2-acetylphenylboronic acid...

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Bibliographic Details
Published in:Chemistry
Main Authors: Bandyopadhyay, Anupam, Gao, Jianmin
Format: Artigo
Language:Inglês
Published: 2015
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC4699557/
https://ncbi.nlm.nih.gov/pubmed/26311464
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/chem.201502077
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