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Modulating Drug Release and Enhancing the Oral Bioavailability of Torcetrapib with Solid Lipid Dispersion Formulations

The development of drug dispersions using solid lipids is a novel formulation strategy that can help address the challenges of poor drug solubility and systemic exposure after oral administration. The highly lipophilic and poorly water-soluble drug torcetrapib could be effectively formulated into so...

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Dettagli Bibliografici
Pubblicato in:AAPS PharmSciTech
Autori principali: Liu, Yajun, Salituro, Gino M., Lee, Keun-joong, Bak, Annette, Leung, Dennis H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer US 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4674632/
https://ncbi.nlm.nih.gov/pubmed/25690735
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12249-015-0299-8
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