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Methadone pharmacogenetics: CYP2B6 polymorphisms determine plasma concentrations, clearance and metabolism

BACKGROUND: Interindividual variability in methadone disposition remains unexplained, and methadone accidental overdose in pain therapy is a significant public health problem. Cytochrome P4502B6 (CYP2B6) is the principle determinant of clinical methadone elimination. The CYP2B6 gene is highly polymo...

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Bibliografski detalji
Izdano u:Anesthesiology
Glavni autori: Kharasch, Evan D., Regina, Karen J., Blood, Jane, Friedel, Christina
Format: Artigo
Jezik:Inglês
Izdano: 2015
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4667947/
https://ncbi.nlm.nih.gov/pubmed/26389554
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1097/ALN.0000000000000867
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