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A Comprehensive in vitro and in silico Analysis of Antibiotics that Activate PXR and Induce CYP3A4 in Liver and Intestine

We have investigated several in silico and in vitro methods in order to improve our ability to predict potential drug interactions of antibiotics. Our focus was to identify those antibiotics that activate PXR and induce CYP3A4 in human hepatocytes and intestinal cells. Human PXR activation was scree...

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Dettagli Bibliografici
Pubblicato in:Drug Metab Dispos
Autori principali: Yasuda, Kazuto, Ranade, Aarati, Venkataramanan, Raman, Strom, Stephen, Chupka, Jonathan, Ekins, Sean, Schuetz, Erin, Bachmann, Kenneth
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2008
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4664062/
https://ncbi.nlm.nih.gov/pubmed/18505790
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.108.020701
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