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Developing a Novel Indolocarbazole as Histone Deacetylases Inhibitor against Leukemia Cell Lines

A novel indolocarbazole (named as ZW2-1) possessing HDAC inhibition activity was synthesized and evaluated against human leukemia cell lines HL-60 and NB4. ZW2-1 performed anti-population growth effect which was in a concentration-dependent manner (2–12 μM) by inducing both apoptosis and autophagy i...

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Pubblicato in:J Anal Methods Chem
Autori principali: Wang, Wenjing, Lv, Maomin, Zhao, Xiong, Zhang, Jingang
Natura: Artigo
Lingua:Inglês
Pubblicazione: Hindawi Publishing Corporation 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4663760/
https://ncbi.nlm.nih.gov/pubmed/26649226
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1155/2015/675053
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