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Lessons from hot spot analysis for fragment-based drug discovery

Analysis of binding energy hot spots at protein surfaces can provide crucial insights into the prospects for successful application of fragment-based drug discovery (FBDD), and whether a fragment hit can be advanced into a high affinity, druglike ligand. The key factor is the strength of the top ran...

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Publicat a:Trends Pharmacol Sci
Autors principals: Hall, David R., Kozakov, Dima, Whitty, Adrian, Vajda, Sandor
Format: Artigo
Idioma:Inglês
Publicat: 2015
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4640985/
https://ncbi.nlm.nih.gov/pubmed/26538314
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tips.2015.08.003
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