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Fluorinated Sterols are Suicide Inhibitors of Ergosterol Biosynthesis and Growth in Trypanosoma brucei

Trypanosoma brucei, the causal agent for sleeping sickness, depends on ergosterol for growth. Herein, we describe the effects of a mechanism-based inhibitor, 26-fluorolanosterol (26FL), which converts in vivo to a fluorinated substrate of the sterol C24-methyltransferase essential for sterol methyla...

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Dettagli Bibliografici
Pubblicato in:Chem Biol
Autori principali: Leaver, David J., Patkar, Presheet, Singha, Ujjial K., Miller, Matthew B., Haubrich, Brad A., Chaudhuri, Minu, Nes, W. David
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4624405/
https://ncbi.nlm.nih.gov/pubmed/26496686
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2015.08.017
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