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Fluorinated Sterols are Suicide Inhibitors of Ergosterol Biosynthesis and Growth in Trypanosoma brucei

Trypanosoma brucei, the causal agent for sleeping sickness, depends on ergosterol for growth. Herein, we describe the effects of a mechanism-based inhibitor, 26-fluorolanosterol (26FL), which converts in vivo to a fluorinated substrate of the sterol C24-methyltransferase essential for sterol methyla...

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Détails bibliographiques
Publié dans:Chem Biol
Auteurs principaux: Leaver, David J., Patkar, Presheet, Singha, Ujjial K., Miller, Matthew B., Haubrich, Brad A., Chaudhuri, Minu, Nes, W. David
Format: Artigo
Langue:Inglês
Publié: 2015
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Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4624405/
https://ncbi.nlm.nih.gov/pubmed/26496686
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2015.08.017
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