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Selective inhibition of PARP10 using a chemical genetics strategy

The lack of inhibitors that are selective for individual poly-ADP-ribose polymerase (PARP) family members has limited our understanding of their roles in cells. Here, we describe a chemical genetics approach for generating selective inhibitors of an engineered variant of PARP10. We synthesized a ser...

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Pubblicato in:Bioorg Med Chem Lett
Autori principali: Morgan, Rory K., Carter-O’Connell, Ian, Cohen, Michael S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4607647/
https://ncbi.nlm.nih.gov/pubmed/26231158
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.07.033
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