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Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP

We previously reported that benzopyrimido-pyrrolo-oxazinedione BPO-27 [6-(5-bromofuran-2-yl)-7,9-dimethyl-8,10-dioxo-11-phenyl-7,8,9,10-tetrahydro-6H-benzo[b]pyrimido [4′,5′:3,4]pyrrolo [1,2-d][1,4]oxazine-2-carboxylic acid] inhibits the cystic fibrosis transmembrane conductance regulator (CFTR) chl...

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Detalhes bibliográficos
Publicado no:Mol Pharmacol
Main Authors: Kim, Yonjung, Anderson, Marc O., Park, Jinhong, Lee, Min Goo, Namkung, Wan, Verkman, A. S.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4576686/
https://ncbi.nlm.nih.gov/pubmed/26174774
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.115.098368
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