Wird geladen...

Optical Isomers of Atorvastatin, Rosuvastatin and Fluvastatin Enantiospecifically Activate Pregnane X Receptor PXR and Induce CYP2A6, CYP2B6 and CYP3A4 in Human Hepatocytes

Atorvastatin, fluvastatin and rosuvastatin are drugs used for treatment of hypercholesterolemia. They cause numerous drug-drug interactions by inhibiting and inducing drug-metabolizing cytochromes P450. These three statins exist in four optical forms, but they are currently used as enantiopure drugs...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Veröffentlicht in:PLoS One
Hauptverfasser: Korhonova, Martina, Doricakova, Aneta, Dvorak, Zdenek
Format: Artigo
Sprache:Inglês
Veröffentlicht: Public Library of Science 2015
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4569258/
https://ncbi.nlm.nih.gov/pubmed/26366873
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0137720
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!