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Differential inhibition of PDKs by phenylbutyrate and enhancement of pyruvate dehydrogenase complex activity by combination with dichloroacetate

Pyruvate dehydrogenase complex (PDHC) is a key enzyme in metabolism linking glycolysis to tricarboxylic acid cycle and its activity is tightly regulated by phosphorylation catalyzed by four pyruvate dehydrogenase kinase (PDK) isoforms. PDKs are pharmacological targets for several human diseases incl...

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Dades bibliogràfiques
Publicat a:J Inherit Metab Dis
Autors principals: Ferriero, Rosa, Iannuzzi, Clara, Manco, Giuseppe, Brunetti-Pierri, Nicola
Format: Artigo
Idioma:Inglês
Publicat: Springer Netherlands 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4551558/
https://ncbi.nlm.nih.gov/pubmed/25601413
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10545-014-9808-2
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