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Differential inhibition of PDKs by phenylbutyrate and enhancement of pyruvate dehydrogenase complex activity by combination with dichloroacetate

Pyruvate dehydrogenase complex (PDHC) is a key enzyme in metabolism linking glycolysis to tricarboxylic acid cycle and its activity is tightly regulated by phosphorylation catalyzed by four pyruvate dehydrogenase kinase (PDK) isoforms. PDKs are pharmacological targets for several human diseases incl...

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Detalhes bibliográficos
Publicado no:J Inherit Metab Dis
Main Authors: Ferriero, Rosa, Iannuzzi, Clara, Manco, Giuseppe, Brunetti-Pierri, Nicola
Formato: Artigo
Idioma:Inglês
Publicado em: Springer Netherlands 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4551558/
https://ncbi.nlm.nih.gov/pubmed/25601413
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10545-014-9808-2
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