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Resin-acid derivatives as potent electrostatic openers of voltage-gated K channels and suppressors of neuronal excitability

Voltage-gated ion channels generate cellular excitability, cause diseases when mutated, and act as drug targets in hyperexcitability diseases, such as epilepsy, cardiac arrhythmia and pain. Unfortunately, many patients do not satisfactorily respond to the present-day drugs. We found that the natural...

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Podrobná bibliografie
Vydáno v:Sci Rep
Hlavní autoři: Ottosson, Nina E, Wu, Xiongyu, Nolting, Andreas, Karlsson, Urban, Lund, Per-Eric, Ruda, Katinka, Svensson, Stefan, Konradsson, Peter, Elinder, Fredrik
Médium: Artigo
Jazyk:Inglês
Vydáno: Nature Publishing Group 2015
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4547393/
https://ncbi.nlm.nih.gov/pubmed/26299574
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep13278
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