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Resin-acid derivatives as potent electrostatic openers of voltage-gated K channels and suppressors of neuronal excitability

Voltage-gated ion channels generate cellular excitability, cause diseases when mutated, and act as drug targets in hyperexcitability diseases, such as epilepsy, cardiac arrhythmia and pain. Unfortunately, many patients do not satisfactorily respond to the present-day drugs. We found that the natural...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Ottosson, Nina E, Wu, Xiongyu, Nolting, Andreas, Karlsson, Urban, Lund, Per-Eric, Ruda, Katinka, Svensson, Stefan, Konradsson, Peter, Elinder, Fredrik
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4547393/
https://ncbi.nlm.nih.gov/pubmed/26299574
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/srep13278
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