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One Crystal, Two Temperatures: Cryocooling Penalties Alter Ligand Binding to Transient Protein Sites

Interrogating fragment libraries by X-ray crystallography is a powerful strategy for discovering allosteric ligands for protein targets. Cryocooling of crystals should theoretically increase the fraction of occupied binding sites and decrease radiation damage. However, it might also perturb protein...

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Detalles Bibliográficos
Publicado en:Chembiochem
Main Authors: Fischer, Marcus, Shoichet, Brian K, Fraser, James S
Formato: Artigo
Idioma:Inglês
Publicado: WILEY-VCH Verlag 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4539595/
https://ncbi.nlm.nih.gov/pubmed/26032594
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201500196
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