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One Crystal, Two Temperatures: Cryocooling Penalties Alter Ligand Binding to Transient Protein Sites

Interrogating fragment libraries by X-ray crystallography is a powerful strategy for discovering allosteric ligands for protein targets. Cryocooling of crystals should theoretically increase the fraction of occupied binding sites and decrease radiation damage. However, it might also perturb protein...

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Pubblicato in:Chembiochem
Autori principali: Fischer, Marcus, Shoichet, Brian K, Fraser, James S
Natura: Artigo
Lingua:Inglês
Pubblicazione: WILEY-VCH Verlag 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4539595/
https://ncbi.nlm.nih.gov/pubmed/26032594
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201500196
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