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One Crystal, Two Temperatures: Cryocooling Penalties Alter Ligand Binding to Transient Protein Sites

Interrogating fragment libraries by X-ray crystallography is a powerful strategy for discovering allosteric ligands for protein targets. Cryocooling of crystals should theoretically increase the fraction of occupied binding sites and decrease radiation damage. However, it might also perturb protein...

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Bibliografiske detaljer
Udgivet i:Chembiochem
Main Authors: Fischer, Marcus, Shoichet, Brian K, Fraser, James S
Format: Artigo
Sprog:Inglês
Udgivet: WILEY-VCH Verlag 2015
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4539595/
https://ncbi.nlm.nih.gov/pubmed/26032594
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201500196
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