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The incorporation of protein flexibility and conformational energy penalties in docking screens to improve ligand discovery

Proteins fluctuate between alternative conformations, which presents a challenge for ligand discovery because such flexibility is difficult to treat computationally owing to problems with conformational sampling and energy weighting. Here, we describe a flexible-docking method that samples and weigh...

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Main Authors: Fischer, Marcus, Coleman, Ryan G., Fraser, James S., Shoichet, Brian K.
Format: Artigo
Sprog:Inglês
Udgivet: 2014
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4144196/
https://ncbi.nlm.nih.gov/pubmed/24950326
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchem.1954
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