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Action potentials and amphetamine release antipsychotic drug from dopamine neuron synaptic VMAT vesicles
Based on lysotracker red imaging in cultured hippocampal neurons, antipsychotic drugs (APDs) were proposed to accumulate in synaptic vesicles by acidic trapping and to be released in response to action potentials. Because many APDs are dopamine (DA) D2 receptor (D2R) antagonists, such a mechanism wo...
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| Опубликовано в: : | Proc Natl Acad Sci U S A |
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| Главные авторы: | , , |
| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
National Academy of Sciences
2015
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4538645/ https://ncbi.nlm.nih.gov/pubmed/26216995 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1503766112 |
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