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Structural Basis for Small Molecule NDB (N-Benzyl-N-(3-(tert-butyl)-4-hydroxyphenyl)-2,6-dichloro-4-(dimethylamino) Benzamide) as a Selective Antagonist of Farnesoid X Receptor α (FXRα) in Stabilizing the Homodimerization of the Receptor

Farnesoid X receptor α (FXRα) as a bile acid sensor plays potent roles in multiple metabolic processes, and its antagonist has recently revealed special interests in the treatment of metabolic disorders, although the underlying mechanisms still remain unclear. Here, we identified that the small mole...

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Détails bibliographiques
Publié dans:J Biol Chem
Auteurs principaux: Xu, Xing, Xu, Xin, Liu, Peng, Zhu, Zhi-yuan, Chen, Jing, Fu, Hai-an, Chen, Li-li, Hu, Li-hong, Shen, Xu
Format: Artigo
Langue:Inglês
Publié: American Society for Biochemistry and Molecular Biology 2015
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4528148/
https://ncbi.nlm.nih.gov/pubmed/26100621
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M114.630475
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