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Direct Coupling of a Seven-Transmembrane-Span Receptor to a Gαi G-Protein Regulatory Motif Complex

Group II activator of G-protein signaling (AGS) proteins contain one or more G-protein regulatory motifs (GPR), which serve as docking sites for Gαi(GDP) independent of Gβγ and stabilize the GDP-bound conformation of Gαi, acting as guanine nucleotide dissociation inhibitors. The GαGPR interaction is...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Mol Pharmacol
Egile Nagusiak: Robichaux, William G., Oner, Sukru S., Lanier, Stephen M., Blumer, Joe B.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: The American Society for Pharmacology and Experimental Therapeutics 2015
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4518091/
https://ncbi.nlm.nih.gov/pubmed/25972449
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.115.097741
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