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Hybrid macrocycle formation and spiro annulation on cis-syn-cis-tricyclo[6.3.0.0(2,6)]undeca-3,11-dione and its congeners via ring-closing metathesis

We have developed a simple methodology to transform cis-syn-cis-triquinane derivative 2 into the diindole based macrocycle 6 involving Fischer indolization and ring-closing metathesis (RCM). Various spiro-polyquinane derivatives have been assembled via RCM as a key step.

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Beilstein J Org Chem
Egile Nagusiak: Kotha, Sambasivarao, Chinnam, Ajay Kumar, Ali, Rashid
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Beilstein-Institut 2015
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4505178/
https://ncbi.nlm.nih.gov/pubmed/26199668
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.11.126
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