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Molecular Dynamics Study of HIV-1 RT-DNA-Nevirapine Complexes Explains NNRTI Inhibition, and Resistance by Connection Mutations

HIV-1 reverse transcriptase (RT) is a multifunctional enzyme that is targeted by nucleoside analogs (NRTIs) and nonnucleoside inhibitors (NNRTIs). NNRTIs are allosteric inhibitors of RT, and constitute an integral part of the highly active antiretroviral therapy (HAART) regimen. Under selective pres...

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Dettagli Bibliografici
Pubblicato in:Proteins
Autori principali: Vijayan, R.S.K., Arnold, Eddy, Das, Kalyan
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4502926/
https://ncbi.nlm.nih.gov/pubmed/24174331
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prot.24460
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