Wordt geladen...

C-Linker Accounts for Differential Sensitivity of ERG1 and ERG2 K(+) Channels to RPR260243-Induced Slow Deactivation

Compounds can activate human ether-à-go-go–related gene 1 (hERG1) channels by several different mechanisms, including a slowing of deactivation, an increase in single channel open probability, or a reduction in C-type inactivation. The first hERG1 activator to be discovered, RPR260243 ((3R,4R)-4-[3-...

Volledige beschrijving

Bewaard in:
Bibliografische gegevens
Gepubliceerd in:Mol Pharmacol
Hoofdauteurs: Gardner, Alison, Sanguinetti, Michael C.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: The American Society for Pharmacology and Experimental Therapeutics 2015
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4468633/
https://ncbi.nlm.nih.gov/pubmed/25888115
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.115.098384
Tags: Voeg label toe
Geen labels, Wees de eerste die dit record labelt!