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Concatenated hERG1 Tetramers Reveal Stoichiometry of Altered Channel Gating by RPR-260243
Activation of human ether-a-go-go–related gene 1 (hERG1) K(+) channels mediates repolarization of action potentials in cardiomyocytes. RPR-260243 [(3R,4R)-4-[3-(6-methoxy-quinolin-4-yl)-3-oxo-propyl]-1-[3-(2,3,5-trifluorophenyl)-prop-2-ynyl]-piperidine-3-carboxylic acid] (RPR) slows deactivation and...
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| Publicado no: | Mol Pharmacol |
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| Main Authors: | , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
The American Society for Pharmacology and Experimental Therapeutics
2015
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4352586/ https://ncbi.nlm.nih.gov/pubmed/25519838 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.114.096693 |
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