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Effects of Ketoconazole on the Pharmacokinetics of Lenvatinib (E7080) in Healthy Participants

BACKGROUND: Lenvatinib is an oral, multitargeted, tyrosine kinase inhibitor under clinical investigation in solid tumors. In vitro evidence indicates that lenvatinib metabolism may be modulated by ketoconazole, an inhibitor of CYP3A4 and p-glycoprotein. METHODS: In this Phase I, single-center, rando...

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Detalhes bibliográficos
Publicado no:Clin Pharmacol Drug Dev
Main Authors: Shumaker, Robert, Aluri, Jagadeesh, Fan, Jean, Martinez, Gresel, Thompson, Gary A, Ren, Min
Formato: Artigo
Idioma:Inglês
Publicado em: BlackWell Publishing Ltd 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4467237/
https://ncbi.nlm.nih.gov/pubmed/26097795
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cpdd.140
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