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Effect of Rifampicin on the Pharmacokinetics of Lenvatinib in Healthy Adults

BACKGROUND AND OBJECTIVES: Lenvatinib is an oral, multitargeted tyrosine kinase inhibitor under clinical investigation in solid tumours. This study evaluated the influence of P-glycoprotein (P-gp) inhibition (single-dose rifampicin) and simultaneous cytochrome P450 3A4 (CYP3A4)/P-gp induction (multi...

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Bibliografiske detaljer
Main Authors: Shumaker, Robert C., Aluri, Jagadeesh, Fan, Jean, Martinez, Gresel, Thompson, Gary A., Ren, Min
Format: Artigo
Sprog:Inglês
Udgivet: Springer International Publishing 2014
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4143598/
https://ncbi.nlm.nih.gov/pubmed/25022720
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40261-014-0217-y
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