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Insights into the slow-onset tight-binding inhibition of Escherichia coli Dihydrofolate Reductase: detailed mechanistic characterization of Pyrrolo [3,2-f] quinazoline-1,3-diamine and its derivatives as novel tight-binding inhibitors

Dihydrofolate reductase, DHFR, is a pivotal enzyme involved in the de novo pathway for purine synthesis, and hence, represents an attractive target to disrupt systems that require rapid DNA turnover. The enzyme acquires resistance to available drugs by various molecular mechanisms, which necessitate...

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Detalhes bibliográficos
Publicado no:FEBS J
Main Authors: Srinivasan, Bharath, Skolnick, Jeffrey
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4445455/
https://ncbi.nlm.nih.gov/pubmed/25703118
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/febs.13244
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