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The Effects of Endoxifen and Other Major Metabolites of Tamoxifen on the Sulfation of Estradiol Catalyzed by Human Cytosolic Sulfotransferases hSULT1E1 and hSULT1A1*1

Tamoxifen is successfully used for both treatment and prevention of estrogen-dependent breast cancer, yet side effects and development of resistance remain problematic. Endoxifen is a major active metabolite of tamoxifen that is being investigated for clinical use. We hypothesized that endoxifen and...

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Veröffentlicht in:Drug Metab Dispos
Hauptverfasser: Squirewell, Edwin J., Duffel, Michael W.
Format: Artigo
Sprache:Inglês
Veröffentlicht: The American Society for Pharmacology and Experimental Therapeutics 2015
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4429681/
https://ncbi.nlm.nih.gov/pubmed/25819444
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.115.063206
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