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Deacetylase inhibitors repress STAT5-mediated transcription by interfering with bromodomain and extra-terminal (BET) protein function

Signal transducer and activator of transcription STAT5 is essential for the regulation of proliferation and survival genes. Its activity is tightly regulated through cytokine signaling and is often upregulated in cancer. We showed previously that the deacetylase inhibitor trichostatin A (TSA) inhibi...

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Dettagli Bibliografici
Pubblicato in:Nucleic Acids Res
Autori principali: Pinz, Sophia, Unser, Samy, Buob, Dominik, Fischer, Philipp, Jobst, Belinda, Rascle, Anne
Natura: Artigo
Lingua:Inglês
Pubblicazione: Oxford University Press 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4402521/
https://ncbi.nlm.nih.gov/pubmed/25769527
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkv188
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