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Deacetylase inhibitors repress STAT5-mediated transcription by interfering with bromodomain and extra-terminal (BET) protein function

Signal transducer and activator of transcription STAT5 is essential for the regulation of proliferation and survival genes. Its activity is tightly regulated through cytokine signaling and is often upregulated in cancer. We showed previously that the deacetylase inhibitor trichostatin A (TSA) inhibi...

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Detaylı Bibliyografya
Yayımlandı:Nucleic Acids Res
Asıl Yazarlar: Pinz, Sophia, Unser, Samy, Buob, Dominik, Fischer, Philipp, Jobst, Belinda, Rascle, Anne
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Oxford University Press 2015
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4402521/
https://ncbi.nlm.nih.gov/pubmed/25769527
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkv188
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