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Deacetylase inhibitors repress STAT5-mediated transcription by interfering with bromodomain and extra-terminal (BET) protein function

Signal transducer and activator of transcription STAT5 is essential for the regulation of proliferation and survival genes. Its activity is tightly regulated through cytokine signaling and is often upregulated in cancer. We showed previously that the deacetylase inhibitor trichostatin A (TSA) inhibi...

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Detalhes bibliográficos
Publicado no:Nucleic Acids Res
Main Authors: Pinz, Sophia, Unser, Samy, Buob, Dominik, Fischer, Philipp, Jobst, Belinda, Rascle, Anne
Formato: Artigo
Idioma:Inglês
Publicado em: Oxford University Press 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4402521/
https://ncbi.nlm.nih.gov/pubmed/25769527
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gkv188
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