Caricamento...

Discovery of a capuramycin analog that kills non-replicating Mycobacterium tuberculosis and its synergistic effects with translocase I inhibitors

Capuramycin (1) and its analogs are strong translocase I (MurX/MraY) inhibitors. In our SAR studies of capuramycin analogs against M. tuberculosis (Mtb), we observed for the first time that a capuramycin analog, UT-01320 (3) killed non-replicating (dormant) Mtb at low concentrations under low-oxygen...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:J Antibiot (Tokyo)
Autori principali: Siricilla, Shajila, Mitachi, Katsuhiko, Wan, Bajoie, Franzblau, Scott G., Kurosu, Michio
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4382465/
https://ncbi.nlm.nih.gov/pubmed/25269459
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/ja.2014.133
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !