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Discovery of a capuramycin analog that kills non-replicating Mycobacterium tuberculosis and its synergistic effects with translocase I inhibitors

Capuramycin (1) and its analogs are strong translocase I (MurX/MraY) inhibitors. In our SAR studies of capuramycin analogs against M. tuberculosis (Mtb), we observed for the first time that a capuramycin analog, UT-01320 (3) killed non-replicating (dormant) Mtb at low concentrations under low-oxygen...

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Dades bibliogràfiques
Publicat a:J Antibiot (Tokyo)
Autors principals: Siricilla, Shajila, Mitachi, Katsuhiko, Wan, Bajoie, Franzblau, Scott G., Kurosu, Michio
Format: Artigo
Idioma:Inglês
Publicat: 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4382465/
https://ncbi.nlm.nih.gov/pubmed/25269459
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/ja.2014.133
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