Φορτώνει......

Phospho-NSAIDs have enhanced efficacy in mice lacking plasma carboxylesterase: Implications for their clinical pharmacology

PURPOSE: The purpose of the study was to evaluate the metabolism, pharmacokinetics and efficacy of phospho-NSAIDs in Ces1c-knockout mice. METHODS: Hydrolysis of phospho-NSAIDs by Ces1c was investigated using Ces1c-overexpressing cells. The rate of phospho-NSAID hydrolysis was compared between wild-t...

Πλήρης περιγραφή

Αποθηκεύτηκε σε:
Λεπτομέρειες βιβλιογραφικής εγγραφής
Τόπος έκδοσης:Pharm Res
Κύριοι συγγραφείς: Wong, Chi C., Cheng, Ka-Wing, Papayannis, Ioannis, Mattheolabakis, George, Huang, Liqun, Xie, Gang, Ouyang, Nengtai, Rigas, Basil
Μορφή: Artigo
Γλώσσα:Inglês
Έκδοση: 2014
Θέματα:
Διαθέσιμο Online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4382427/
https://ncbi.nlm.nih.gov/pubmed/25392229
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-014-1565-2
Ετικέτες: Προσθήκη ετικέτας
Δεν υπάρχουν, Καταχωρήστε ετικέτα πρώτοι!