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Design and Synthesis of Acetylenyl Benzamide Derivatives as Novel Glucokinase Activators for the Treatment of T2DM

[Image: see text] Novel acetylenyl-containing benzamide derivatives were synthesized and screened using an in vitro assay measuring increases in glucokinase activity stimulated by 10 mM glucose concentration and glucose uptake in rat hepatocytes. Lead optimization of an acetylenyl benzamide series l...

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Bibliografiske detaljer
Udgivet i:ACS Med Chem Lett
Main Authors: Park, Kaapjoo, Lee, Byoung Moon, Hyun, Kwan Hoon, Han, Taedong, Lee, Dong Hoon, Choi, Hyun Ho
Format: Artigo
Sprog:Inglês
Udgivet: American Chemical Society 2015
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4360162/
https://ncbi.nlm.nih.gov/pubmed/25815149
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml5004712
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