Načítá se...

Design and Synthesis of Acetylenyl Benzamide Derivatives as Novel Glucokinase Activators for the Treatment of T2DM

[Image: see text] Novel acetylenyl-containing benzamide derivatives were synthesized and screened using an in vitro assay measuring increases in glucokinase activity stimulated by 10 mM glucose concentration and glucose uptake in rat hepatocytes. Lead optimization of an acetylenyl benzamide series l...

Celý popis

Uloženo v:
Podrobná bibliografie
Vydáno v:ACS Med Chem Lett
Hlavní autoři: Park, Kaapjoo, Lee, Byoung Moon, Hyun, Kwan Hoon, Han, Taedong, Lee, Dong Hoon, Choi, Hyun Ho
Médium: Artigo
Jazyk:Inglês
Vydáno: American Chemical Society 2015
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4360162/
https://ncbi.nlm.nih.gov/pubmed/25815149
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml5004712
Tagy: Přidat tag
Žádné tagy, Buďte první, kdo otaguje tento záznam!