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Novel mixed NOP/MOP agonist BU08070 alleviates pain and inhibits gastrointestinal motility in mouse models mimicking diarrhea-predominant irritable bowel syndrome symptoms

BACKGROUND: The opioid and nociceptin systems play a crucial role in the maintenance of homeostasis in the gastrointestinal (GI) tract. The aim of this study was to characterize the effect of BU08070, a novel mixed MOP/NOP agonist, on mouse intestinal contractility in vitro and GI motility in vivo i...

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Detaylı Bibliyografya
Yayımlandı:Eur J Pharmacol
Asıl Yazarlar: Sobczak, Marta, Cami-Kobeci, Gerta, Sałaga, Maciej, Husbands, Stephen M., Fichna, Jakub
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2014
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4341819/
https://ncbi.nlm.nih.gov/pubmed/24815321
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejphar.2014.04.038
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