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Exploring the drug resistance of V32I and M46L mutant HIV-1 protease to inhibitor TMC114: flap dynamics and binding mechanism

Inhibitors of HIV-1 protease (HIV-1-pr) generally only bind to the active site of the protease. However, for some mutants such as V32I and M46L the TMC114 can bind not only to the active cavity also to the groove of the flexible flaps. Although the second binding site suggests the higher efficiency...

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Detalhes bibliográficos
Publicado no:J Mol Graph Model
Main Authors: Meher, Biswa Ranjan, Wang, Yixuan
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4314403/
https://ncbi.nlm.nih.gov/pubmed/25562662
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jmgm.2014.11.003
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