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In Vitro Resistance Selection with Doravirine (MK-1439), a Novel Nonnucleoside Reverse Transcriptase Inhibitor with Distinct Mutation Development Pathways

Doravirine (DOR, formerly known as MK-1439) is a human immunodeficiency type 1 virus (HIV-1) nonnucleoside reverse transcriptase inhibitor (NNRTI) that is currently in phase 2b clinical trials. In vitro resistance selection of subtype B virus (MT4-green fluorescent protein [GFP] cells), as well as s...

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Опубликовано в: :Antimicrob Agents Chemother
Главные авторы: Feng, Meizhen, Wang, Deping, Grobler, Jay A., Hazuda, Daria J., Miller, Michael D., Lai, Ming-Tain
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Microbiology 2014
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4291404/
https://ncbi.nlm.nih.gov/pubmed/25385110
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.04201-14
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