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MMP9-sensitive polymers mediate environmentally-responsive bivalirudin release and thrombin inhibition

MMP9-responsive bivalirudin-HPMA copolymers were synthesized for direct, local administration in rat spinal cord contusion injury models. Polymer-conjugated bivalirudin peptides maintained activity while demonstrating enzyme-mediated release upon MMP9 exposure and prolonged release from hyaluronic a...

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Detalhes bibliográficos
Publicado no:Biomater Sci
Main Authors: Chu, D.S., Sellers, D.L., Bocek, M.J., Fischedick, A.E., Horner, P.J., Pun, S.H.
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4289632/
https://ncbi.nlm.nih.gov/pubmed/25589953
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C4BM00259H
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