Caricamento...

Specific binding of lacosamide to collapsin response mediator protein 2 (CRMP2) and direct impairment of its canonical function: implications for the therapeutic potential of lacosamide

The novel anti-epileptic drug lacosamide (LCM; SPM927, Vimpat(®)) has been heralded as having a dual-mode of action through interactions with both the voltage-gated sodium channel and the neurite outgrowth-promoting collapsin response mediator protein 2 (CRMP2). Lacosamide’s ability to dampen neuron...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Mol Neurobiol
Autori principali: Wilson, Sarah M., Khanna, Rajesh
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4272652/
https://ncbi.nlm.nih.gov/pubmed/24944082
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s12035-014-8775-9
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !