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Crystal Structure of Sphingosine Kinase 1 with PF-543

[Image: see text] The most potent inhibitor of Sphingosine Kinase 1 (SPHK1) so far identified is PF-543. The crystal structure of SPHK1 in complex with inhibitor PF-543 to 1.8 Å resolution reveals the inhibitor bound in a bent conformation analogous to that expected of a bound sphingosine substrate...

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Bibliografski detalji
Izdano u:ACS Med Chem Lett
Glavni autori: Wang, Jing, Knapp, Stefan, Pyne, Nigel J., Pyne, Susan, Elkins, Jonathan M.
Format: Artigo
Jezik:Inglês
Izdano: American Chemical Society 2014
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4265818/
https://ncbi.nlm.nih.gov/pubmed/25516793
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml5004074
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